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邓卫平 教授、博士生导师、副院长
联系方式：
通讯地址：上海市梅陇路130号318信箱，邮编200237
电话：（021）64252431
个人简介：
1995年毕业于浙江师范大学，2000年获中国科学院上海有机化学研究所理学博士学位，导师戴立信院士。2000年至2003年先后在美国国立卫生研究院和美国Rochester大学化学系进行博士后研究。2003年底加入新加坡的新药研发公司---S*BIO，进行靶向小分子抗癌药物的研发工作。2005年8月受聘于华东理工大学药学院。回国先后获得一系列荣誉和称号，包括：上海市浦江人才(2006)，教育部新世纪优秀人才(2007)，上海市育才奖(2007)，华东理工大学优秀教育工作者(2009)，上海市曙光学者(2009)，上海市归侨侨眷先进个人(2010)，华东理工大学育英奖(2010)以及东岳-天鼎奖教金特等奖（2015）等。兼任教育部高等学校药学类专业教学指导委员会（大）药学分委会委员，上海市药学会药物化学专委会委员，中国医药工业杂志编委等职。先后承担国家自然科学基金、上海市基础研究重点项目等十余项研究项目。已在国际核心刊物J. Am. Chem. Soc.; Angew. Chem. Int. Ed.; ACS Catal.; Chem. Commun.; Org. Lett.; Chem. Eur. J. 等上发表100余篇SCI论文和专利申请。译著《药物考》和《创新药物发现-实践、过程和展望》；参编教材《药物化学》双语教材，参编论著Stereoselective synthesis of planar chiral ferrocenes: Chiral Ferrocenes in Asymmetric Catalysis(2010)。
主要研究方向：
1. 基于手性技术的碳碳键及碳杂原子键的形成方法学，以及新型手性催化剂的设计合成及应用研究。
2. 基于新概念，新试剂和新反应的新型杂环化合物的设计合成及其生理活性研究。
3. 化学创新药物及"Me Too"药物的绿色合成技术的开发研究。
4. 基于组蛋白去乙酰化酶（HDAC）抑制剂的靶向小分子抗肿瘤药物研究。
热烈欢迎有志于手性技术和药物发现研究的优秀学子加入我们团队！
代表性论文(2010-)：
2021
102. Zhang Jian, Gao Yan-Shan, Gu Bu-Ming, Yang Wu-Lin, Tian Bo-Xue, Deng Wei-Ping. Cooperative N-heterocyclic Carbene and Iridium Catalysis Enables Stereoselective and Regiodivergent [3+2] and [3+3] Annulation Reactions. ACS Catal., 2021, 11, 3810-3821.
101. Yang Wu-Lin, Liu Tian-Tian, Ni Tao, Zhu Bin, Luo Xiaoyan, Deng Wei-Ping. Iridium-Catalyzed Asymmetric Cascade Allylation/Pictet-Spengler Cyclization Reaction for the Enantioselective Synthesis of 1,3,4-Trisubstituted Tetrahydroisoquinolines. Org. Lett., 2021, 23, DOI: 10.1021/acs.orglett.1c00709.
100. Liu Yang-Zi, Wang Zhongao, Huang Zesheng, Yang Wu-Lin, Deng Wei-Ping.Sulfone as a Transient Activating Group in the Palladium-Catalyzed Asymmetric [4 + 3] Cycloaddition of Trimethylenemethane Enabling the Enantioselective Synthesis of Fused Azepines. Org. Lett., 2021, 23, 588-594.
99. Yang Wu-Lin, Ni Tao, Deng Wei-Ping. Iridium-Catalyzed Diastereo- and Enantioselective [4 + 3] Cycloaddition of 4‑Indolyl Allylic Alcohols with Azomethine Ylides. Org. Lett., 2021, 23, 588-594.
98. Tian Fei, Yang Wu-Lin, Ni Tao, Zhang Jian, Deng Wei-Ping. Catalytic asymmetric dipolar cycloadditions of indolyl delocalized metal-allyl species for the enantioselective synthesis of cyclopenta[b]indoles and pyrrolo[1,2-a] indoles. Sci. Chin. Chem., 2021, 64(1), 34-40.
97. Xu Hui, Han Teng, Luo Xiaoyan, Deng Wei-Ping. The construction of 3-azabicyclo[3.1.0]hexane backbone by the reaction of allenes with allylamines via tandem aza-Michael addition and Copper-mediated oxidative carbanion cyclization. Chin. J. Chem., 2021, 39, 666-670.
2020
96. Liu Yang-Zi, Wang Zhongao, Huang Zesheng, Zheng Xing, Yang Wu-Lin, Deng Wei-Ping. Palladium-Catalyzed Asymmetric [4 + 3] Cyclization of Trimethylenemethane: Regio-, Diastereo-, and Enantioselective Construction of Benzofuro[3,2-b]azepine Skeletons. Angew. Chem. Int. Ed., 2020, 59, 1238-1242.
95. Zhang Jian, Ni Tao, Yang Wu-Lin, Deng Wei-Ping. Catalytic Asymmetric [3 + 2] Annulation via Indolyl Copper-Allenyliende Intermediates: Diastereo- and Enantioselective Assembly of Pyrrolo[1,2-a]indoles. Org. Lett., 2020, 22, 4547-4552.
94. Deng Hua, Liu Tian-Tian, Ding Zheng-Dong, Yang Wu-Lin, Luo Xiaoyan, Deng Wei-Ping. Kinetic resolution of 2H-azirines via Cu(I)-catalyzed asymmetric 1,3-dipolar cycloaddition of azomethine ylides. Org. Chem. Front., 2020, 7(20), 3247-3252.
93. Ye Chao, Yang Wu-Lin, Zhai Yufei, Deng Hua, Luo Xiaoyan, Kai Guoyin, Deng Wei-Ping. Copper(I)-Catalyzed Asymmetric [3 + 3] Annulation Involving Aziridines to Construct Tetrahydro-β-carbolines. Org. Chem. Front., 2020, 7(21), 3393-3398
92. Ding Xiang-Feng, Deng Wei-Ping. Asymmetric Inverse-Electron-Demand Diels-Alder Reaction of 2-Pyrones. Chin. J. Org. Chem., 2020, 40, 3976-3977. (Highlight)
91. Yang Wu-Lin, Huang Zesheng, Liu Yang-Zi, Yu Xingxin, Deng Wei-Ping. Highly Regio-, Diastereo-, and Enantioselective Assembly of Azepino[2,3‑b]indoles via Palladium-Catalyzed [4 + 3] Cycloaddition. Chin. J. Chem., 2020, 38(12), 1571-1574.
90. Tian Fei, Zhang Jian, Yang Wu-Lin, Deng Wei-Ping. Progress in Iridium-Catalyzed Asymmetric Allylic Substitution Reactions via Synergetic Catalysis. Chin. J. Org. Chem., 2020, 40, 3262-3278.
89. Yang Wu-Lin, Li Wen, Yang Zhong-Tao, Deng Wei-Ping. Organocatalytic Regiodivergent Ring Expansion of Cyclobutanones for the Enantioselective Synthesis of Azepino[1,2‑a]indoles and Cyclohepta[b]indoles. Org. Lett. 2020, 22, 4026-4032.
88. Zou Xue-Jie, Yang Wu-Lin, Zhu Jing-Yan, Deng Wei-Ping. Catalytic Enantioselective Formal Synthesis of MDM2 Antagonist RG7388 and Its Analogue. Chin. J. Chem., 2020, 38(5), 435-438.
87. Zheng Xing, Sun Hao, Yang Wu-Lin, Deng Wei-Ping. Elaboration of phosphoramidite ligands enabling palladium-catalyzed diastereo- and enantioselective all carbon [4+3] cycloaddition. Sci. Chin. Chem., 2020, 63, 911-916.
86. Zou Xuejie, Liu Yangzi, Shang Shaojing, Yang Wulin, Deng Wei-Ping. Diastereoselective Synthesis of Functional ized Tetrahydro-γ-Carbolines via a [3+3] Cycloaddition of 2,2'-Diester Aziridines with β-(Indol-2-yl)-α,β-unsaturated Ketones. Chin. Chem. Lett., 2020, 31, 1293-1296.
85. Yang Wulin, Wang Hao, Pan Zirong, Li Zhong, Deng Wei-Ping. Asymmetric synthesis of pyrrolo[1,2-a]indoles via organocatalytic[3+2] annulation of substituted 2-vinylindoles with azlactones. Chin. Chem. Lett., 2020, 31, 721-724.
2019
84. Leng Jiaying, Xu Hui, Meng Jiang, Luo Xiaoyan, Deng Wei-Ping. Transition-metal-free synthesis of polysubstituted pyrrole derivatives via [4+1] annulation of beta-keto acids (C1 synthon) and alpha,beta-unsaturated imines. Tetrahedron, 2019, 75, 130709.
83. Zhu Jinbin, Huang Linwei, Dong Wei, Li Naikai, Yu Xingxin, Deng Wei-Ping, Tang Wenjun. Enantioselective Rhodium-Catalyzed Addition of Arylboroxines to N-Unprotected Ketimines: Efficient Synthesis of Cipargamin. Angew. Chem. Int. Ed., 2019, 58, 16119-16123. (VIP)
82. Chen Long, Yang Wu-Lin, Shen Jia-Huan, Deng Wei-Ping. Nickel(II)-Catalyzed Diastereo- and Enantioselective Michael/Hemiacetalization Cascade Reaction of α-Ketoesters with 2-(2-Nitrovinyl)phenols. Adv. Synth. Catal., 2019, 361(19), 4611-4622.
81. Mao Jia, Zhang Hao, Ding Xiang-Feng, Luo Xiaoyan, Deng Wei-Ping. Synergistic Catalysis for Asymmetric [3 + 2] Cycloadditions of 2-Indolylmethanols with α,β-Unsaturated Aldehydes. J. Org. Chem. 2019, 84(17), 11186-11194.
80. Wu Shu-Xiao, Gu Bo-Qi, Xu Hui, Zheng Xing, Luo Xiaoyan, Deng Wei-Ping. Organocatalytic Asymmetric Inverse-Electron-Demand Diels-Alder Reaction of Pyrrolidone-Dienes with Enals. Adv. Synth. Catal., 2019, 361(18), 4302-4313.
79. Deng Hua, Jia Renmeng, Yang Wu-Lin, Yu Xingxin, Deng Wei-Ping. Ligand-Controlled Switch in Diastereoselectivities: Catalytic Asymmetric Construction of Spirocyclic Pyrrolidine-azetidine/oxe(thie)tane Derivatives. Chem. Commun., 2019, 55, 7346-7349.
78. Ding Xiang-Feng, Yang Wu-Lin, Mao Jia, Cao Cong-Xian, Deng Wei-Ping. Enantioselective Construction of Dihydropyrido[1,2-a]indoles via Organocatalytic Arylmethylation of 2-Enals with Inert Aryl Methane Nucleophiles. Org. Lett., 2019, 21, 5514-5518.
77. Jin Jing-Hai, Zhao Jianhong, Yang Wu-Lin, Deng Wei-Ping. Asymmetric synthesis of spirooxindole β-lactams via isothiourea-catalyzed Mannich/lactamization reaction of aryl acetic acids with isatin-derived ketimines. Adv. Synth. Catal., 2019, 361(7), 1592-1596.
76. Yang Zhong-Tao, Zhao Jianhong, Yang Wu-Lin, Deng Wei-Ping. Enantioselective Construction of CF3‑Containing Spirooxindole γ‑Lactones via Organocatalytic Asymmetric Michael/Lactonization. Org. Lett., 2019, 21, 1015-1020.
75. Yang Wu-Lin, Sun Zhong-Tao, Sun Hao, Deng Wei-Ping. Nickel(II)-Catalyzed Diastereo- and Enantioselective [3+2] Cycloaddition of α-Ketoesters with 2-Nitrovinylindoles and 2-Nitrovinylpyrroles. Chin. J. Chem., 2019, 37, 216-220.
74. Yang Wu-Lin, Sun Zhong-Tao, Zhang Jian, Li Zhong, Deng Wei-Ping. Enantioselective synthesis of 3-amino-hydrobenzofuran-2,5-diones via Cu(I)-catalyzed intramolecular conjugate addition of imino esters. Org. Chem. Front., 2019, 6, 579-583.
2018
73. Gu Bo-Qi, Yang Wu-Lin, Wu Shu-Xiao, Wang Yan-Bing, Deng Wei-Ping. Organocatalytic asymmetric synthesis oftetrahydrocarbazoles via an inverse-electron demand Diels–Alder reaction of 2,3-indole-dieneswith enals. Org. Chem. Front., 2018, 5, 3430-3434.
72. Leng Jiaying, Meng Jiang, Luo Xiaoyan, Deng Wei-Ping. Formal [4 + 1] Cycloaddition Strategy for the Synthesis of Dihydrobenzofurans via Michael Addition of 2-(2-nitrovinyl)-phenols and Malonate Esters (C1 Synthon) and Subsequent Iodine-catalyzed Oxidative Annulation. Tetrahedron, 2018, 74, 6993-6999.
71. Jin Jing-Hai, Li Xiang-Yu, Luo Xiaoyan, Deng Wei-Ping. Enantioselective synthesis of indolo[2,3-b]-dihydrothiopyranones via [3+3] cycloaddition of chiral α,β-unsaturated acylammonium salts. Tetrahedron, 2018, 74, 6804-6808.(Highlighted by Synfacts 2019, 15(02), 0132.)
70. Ding Xiang-Feng, Su Ruo-Heng, Yang Wu-Lin, Deng Wei-Ping. Organocatalytic Asymmetric Formal Aza-[3 + 3] Cycloadditions of 3-Aminobenzofuran with α,β-Unsaturated Aldehydes. Adv. Synth. Catal., 2018, 360, 4168-4177.
69. Deng Hua, Yang Wu-Lin, Tian Fei, Tang Wenjun, Deng Wei-Ping. Asymmetric Construction of 3-Azabicyclo[3.1.0]hexane Skeleton with Five Contiguous Stereogenic Centers by Cu-Catalyzed 1,3-Dipolar Cycloaddition of Trisubstituted Cyclopropenes. Org. Lett., 2018, 20(13), 4121-4125. (Highlighted by Synfacts 2018, 14(9), 0935.)
68. Tian Fei, He Fu-Sheng, Deng Hua, Yang Wu-Lin, Deng Wei-Ping. β-Silyl Acrylates in Asymmetric [3 + 2] Cycloadditions Affording Pyrrolidine Azasugar Derivatives. Org. Lett., 2018, 20(13), 3838-3842. (Highlighted by Synfacts 2018, 14(9), 0936.)
67. Zheng Xing, Yang Wu-Lin, Liu Yang-Zi, Wu Shu-Xiao, Deng Wei-Ping. Enantioselective Synthesis of Tropanes via [3+3] Annulation of Cyclic Azomethine Ylides with Substituted 2-Vinylindoles and 2-Vinylpyrroles. Adv. Synth. Catal., 2018, 360(15), 2843-2853.(VIP) (Highlighted by Synfacts 2018, 14(8), 0846.)
66. Liu Yang-Zi, Shang Shao-Jing, Zhu Jing-Yan, Yang Wu-Lin, Deng Wei-Ping. Regioselective and Stereoselective [3 + 3] Annulation of Ketones Derived Azomethine Ylides with 2-Indolylethylenes: Direct Access to Highly Substituted Tetrahydro-γ-Carbolines. Adv. Synth. Catal., 2018, 360(11), 2191-2203.
65. Zhu Jing-Yan, Yang Wu-Lin, Liu Yang-Zi, Shang Shao-Jing, Deng Wei-Ping. Copper(I)-catalyzed Asymmetric Mannich Reaction of Glycine Schiff Bases with Isatin-derived Ketimines: Enantioselective Synthesis of 3-Substituted 3-Aminooxindoles. Org. Chem. Front., 2018, 5, 70-74.
64. Jin Jing-Hai, Wang Hao, Yang Zhong-Tao, Yang Wu-Lin, Tang Wenjun, Deng Wei-Ping. Asymmetric Synthesis of 3,4-Dihydroquinolin-2-ones via a Stereoselective Palladium-Catalyzed Decarboxylative [4 + 2] Cycloaddition. Org. Lett., 2018, 20(1), 104-107. (Highlighted by Synfacts 2018, 14(3), 0288.)
63. Han Teng, Wang Yu, Li Hong-Liang, Luo Xiaoyan, Deng Wei-Ping. Synthesis of Polysubstituted 3-Aminothiophenes from Thioamides and Allenes via Tandem Thio-Michael Addition/Oxidative Annulation and 1,2-Sulfur Migration. J. Org. Chem., 2018, 83, 1538-1542.
62. Jia Renmeng, Meng Jiang, Leng Jiaying, Yu Xingxin, Deng Wei-Ping. Rhodium(II)-Catalyzed Reaction of 1‑Tosyl-1,2,3-triazoles with Morita–Baylis–Hillman adducts: Synthesis of 3,4-Fused Pyrroles. Chem. Asian J., 2018, 13, 2360-2364.
61. Yang Zhong-Tao, Yang Wu-Lin, Chen Long, Sun Hao, Deng Wei-Ping. Organocatalytic Enantioselective aza-Friedel-Crafts Reactions of Pyrazolinone Ketimines with Hydroxyindoles and Electron-Rich Phenols. Adv. Synth. Catal., 2018, 360(10), 2049-2054.
60. Wen Min, Sun Pei-Pei, Luo Xiaoyan, Deng Wei-Ping. Cu(II)-catalyzed one-pot synthesis of fully substituted dihydrothiophenes and thiophenes from thioamides and enynones. Tetrahedron, 2018, 74(31), 4168-4173.
2017
59. He Fu-Sheng, Li Cong-Shan, Deng Hua, Zheng Xing, Yang Zhong-Tao, Deng Wei-Ping. The facile and stereoselective synthesis of pyrrolidine β-amino acids via copper(I)-catalyzed asymmetric 1,3-dipolar cycloaddition. Org. Chem. Front., 2017, 4, 52-56.
58. Liu Yang-Zi, Shang Shao-Jing, Yang Wu-Lin, Luo Xiaoyan, Deng Wei-Ping. Stereoselective Synthesis of Pyrrolidines Containing a 3‑Fluoro Quaternary Stereocenter via Copper(I)-Catalyzed Asymmetric 1,3-Dipolar Cycloaddition. J. Org. Chem., 2017, 82(20), 11141-11149.
57. Jin Jing-Hai, Xu Qin-Chang, Deng Wei-Ping. DMAP-catalyzed [4+2] cycloaddition of α,β-unsaturated carboxylic acids with ketones for the synthesis of α,β-unsaturated δ-lactones. Chin. J. Chem., 2017, 35, 397-400.
56. Meng Jiang, Wen Min, Zhang Shiwei, Pan Peiwen, Yu Xingxin, Deng Wei-Ping. Unexpected O-H Insertion of Rhodium-Azavinylcarbenes with N-Acylhydrazones: Divergent Synthesis of 3,6-Disubstituted and 3,5,6-Trisubstituted-1,2,4-Triazines. J. Org. Chem., 2017, 82, 1676-1687. (Highlighted by Synfacts 2017, 13(4), 0354.)
55. Jin Jing-Hai, Li Xiang-Yu, Luo Xiaoyan, Fossey John S., Deng Wei-Ping. Asymmetric Synthesis of cis-3,4-Dihydrocoumarins via [4 + 2] Cycloadditions Catalyzed by Amidine Derivatives. J. Org. Chem., 2017, 82, 5424-5432.
54. Meng Jiang, Jia Renmeng, Leng Jiaying, Wen Min, Yu Xingxin, Deng Wei-Ping. Carbon-Carbon Bond Formation by Reaction of Rhodium Azavinylcarbenes with Secondary Amides: Access to Indigo Analogues from Isatins. Org. Lett., 2017, 19, 4520-4523.
53. Deng Hua, He Fu-Sheng, Li, Cong-Shan, Deng Wei-Ping. Enantioselective Construction of Tricyclic Pyrrolidine-Fused Benzo[b]thiophene 1,1-Dioxides Derivatives via Copper(I)-Catalyzed Asymmetric 1,3-Dipolar Cycloaddition. Org. Chem. Front., 2017, 4, 2343-2347.
52. Su Ruo-Heng, Ding Xiang-Feng, Wu Shu-Xiao, Zhao Jian-Hong, Deng Wei-Ping. Secondary Amine-catalyzed Asymmetric Formal Aza [3+3] Cycloaddition to Construct Enantioenriched Piperidines Derivatives. Tetrahedron, 2017, 73(41), 6031-6038.
2016
51. He Fu-Sheng, Jin Jing-Hai, Yang Zhong-Tao, Yu Xingxin, Fossey John S., Deng Wei-Ping. Direct Asymmetric Synthesis of β-Bis-Aryl-α-Amino Acid Esters via Enantioselective Copper-Catalyzed Addition of p-Quinone Methides. ACS Catalysis, 2016, 6(2), 652-656. (Highlighted by Synfacts 2016, 12(4), 0390.)
50. Huang Linwei, Zhu Jinbin, Jiao Guangjun, Wang Zheng, Yu Xingxin, Deng Wei-Ping, Tang Wenjun. Highly Enantioselective Rhodium-Catalyzed Addition of Arylboroxines to Simple Aryl Ketones: Efficient Synthesis of Escitalopram. Angew. Chem. Int. Ed., 2016, 55(14), 4527-4531. (Highlighted by Synfacts, 2016, 12(6), 0557.)
49. Li Hong-Liang, Wang Yu, Sun Pei-Pei, Luo Xiaoyan, Shen Zhenlu, Deng Wei-Ping. α,β-Double electrophilic addition of allene-1,3-dicarboxylic esters for the construction of polysubstituted furans via KI/TBHP promoted oxidative annulation. Chem. Eur. J., 2016, 22, 9348-9355.
48. Yang Wu-Lin, Li Chun-Yan, Qin Wen-Jing, Tang Fei-Fei, Yu Xingxin, Deng Wei-Ping. Cu(I)-Catalyzed Chemoselective and Stereoselective [3 + 3] Cycloaddition of Azomethine Ylides with 2-Indolylnitroethylenes: Facile Access to Highly Substituted Tetrahydro-γ-Carbolines. ACS Catalysis, 2016, 6, 5685-5690. (Highlighted by Synfacts, 2016, 12(10), 1058.)
47. Wang Yu, Jiang Chen-Min, Li Hong-Liang, He Fu-Sheng, Luo Xiaoyan, Deng Wei-Ping. Regioselective Iodine-catalyzed Construction of Polysubstituted Pyrroles from Allenes and Enamines. J. Org. Chem., 2016, 81, 8653-8658.
46. Gu Bo-Qi, Zhang Hao, Su Ruo-Heng, Deng Wei-Ping. Organocatalytic asymmetric synthesis of dihydrocarbazoles via a formal [4+2] cycloaddition of in situ generated o-quinodimethanes with enals. Tetrahedron, 2016, 72, 6595-6602.
45. Zhu Mingyu, Deng Weiping. An-PIQ Catalyzed Kinetic Resolution of β-Iodo Morita–Baylis–Hillman Adducts. Chin. J. Org. Chem., 2016, 36 (10): 2397-2406.
44. Li Hongliang, Wang Zhenglin, Deng Weiping. Cu(I)-Catalyzed Intramolecular Cyclization of Ortho-halogenated Phenylthioacetamides for the Synthesis of 2-Amino Benzo[b]thiophenes. Chin. J. Org. Chem., 2016, 36 (10): 2419-2425.
43. Meng Jiang, Ding Xiangfeng, Yu Xingxin, Deng Wei-Ping. Synthesis of 2,5-epoxy-1,4-benzoxazepines via rhodium(II)-catalyzed reaction of 1-tosyl-1,2,3- triazoles and salicylaldehydes. Tetrahedron, 2016, 72, 176-183.
2015
42. Jiang Shan-Shan, Xu Qin-Chang, Zhu Ming-Yu, Yu Xingxin, Deng Wei-Ping. Kinetic Resolution of α-Methylene-β-hydroxy Esters Catalyzed by Acyl Transfer Catalyst An-PIQ. J. Org. Chem., 2015, 80, 3159-3169.
41. Jiang Shan-Shan, Gu Bo-Qi, Zhu Ming-Yu, Yu Xingxin, Deng Wei-Ping. Nonenzymatic kinetic resolution of α-aryl substituted allylic alcohols catalyzed by acyl transfer catalyst Np-PIQ. Tetrahedron, 2015, 71, 1187-1191.
40. Qin Wen-Jing, Li Yi, Yu Xingxin, Deng Wei-Ping. TBAI/TBHP catalyzed direct N-acylation of sulfoximines with aldehydes. Tetrahedron, 2015, 71, 1182-1186.
39. Li Hong-Liang, An Xing-Lan, Ge Li-Shi, Luo Xiaoyan, Deng Wei-Ping. Catalyitc α-Hydroxylation of Ketones under CuBr2 or HBr/DMSO Systems. Tetrahedron, 2015, 71, 3247-3252.
38. Meng Jiang, Wu Di, Shi Ying, Yu Xingxin, Deng Wei-Ping. Construction of 1H-pyrrol-2-ylphosphonates via [3+2] cycloaddition of phosphate azomethine ylides with ynones. Tetrahedron, 2015, 71, 1074-1079.
37. Luo Xiaoyan, Ge Li-Shi, An Xing-Lan, Jin Jing-Hai, Wang Yu, Sun Pei-Pei, Deng Wei-Ping. Regioselective Metal-Free One-pot Synthesis of Functionalized 2-Aminothiophene Derivatives. J. Org. Chem., 2015, 80, 4611-4617.
36. Yang Wu-Lin, Liu Yang-Zhi, Luo Shuai, Yu Xingxin, Fossey John S., Deng Wei-Ping. Copper-catalyzed asymmetric construction of dispiropyrrolidine skeleton via 1,3-dipolarcycloaddition of azomethine ylides with α-alkylidene. Chem. Commun., 2015, 51, 9212-9215. (Highlighted by Synfacts, 2015, 11(12), 738.)
35. Wang Zheng, Yu Xingxin, Tian Bo-Xue, Payne Daniel T., Yang Wu-Lin, Liu Yang-Zi, Fossey John S., Deng Wei-Ping. Chiral N,O-Ligand/Cu(OAc)2 Catalyzed Asymmetric Construction of 4-Aminopyrrolidine Derivatives via 1,3-Dipolar Cycloaddition of Azomethine Ylides with α-phthalimidoacrylates. Chem. Eur. J., 2015, 21, 10457-10465.
34. Tang Fei-Fei, Yang Wu-Lin, Yu Xingxin, Deng Wei-Ping. Cu(OAc)2/FOXAP complex catalyzed construction of 2,5-dihydropyrrole derivatives via asymmetric 1,3-dipolar cycloaddition of azomethine ylides with ethynyl ketones. Catal. Sci. Technol., 2015, 5, 3568-3575.
33. Yang Wu-Lin, Tang Fei-Fei, He Fu-Sheng, Li Chun-Yan, Yu Xingxin, Deng Wei-Ping. Asymmetric construction of spirocyclic pyrrolidine- thia(oxa)zolidinediones via N,O-ligand/Cu(I) catalyzed 1,3-dipolar cycloaddition of azomethine ylides with 5-alkylidene thia(oxa)zolidine-2,4-diones. Org. Lett., 2015, 17, 4822-4825. (Highlighted by Synfacts, 2015, 11(12), 1285.)
32. He Fu-Sheng, Zhu Han, Wang Zheng, Gao Ming, Yu Xingxin, Deng Wei-Ping. Asymmetric Construction of 3,4-Diamino Pyrrolidines via Chiral N,O-Ligand/Cu(I) Catalyzed 1,3-Dipolar Cycloaddition of Azomethine Ylides with β‑Phthalimidonitroethene. Org. Lett., 2015, 17, 4988-4991. (Highlighted by Synfacts 2015, 11(12), 1284.)
31. Li Chun-Yan, Yang Wu-Lin, Luo Xiaoyan, Deng Wei-Ping. Diastereodivergent asymmetric Michael addition of cyclic azomethine ylides to nitroalkenes: direct approach for the synthesis of 1,7-diazaspiro[4.4]nonane diastereoisomers. Chem. Eur. J., 2015, 21, 19048-19057. (Highlighted by Synfacts 2016, 12(2), 0167.)
2014
30. Wang Zheng, Ye Jinjin, Wu Rui, Liu Yang-Zi, Fossey John S., Cheng Jiagao, Deng Wei-Ping. Bi-Aryl Rotation in Phenyl-dihydroimidazoquinoline Catalysts for Kinetic Resolution of Arylalkyl Carbinols. Catal. Sci. Technol., 2014, 4 (7), 1909-1913.
29. Wang Zheng-Lin, Li Hong-Liang, Ge Li-Shi, An Xing-Lan, Zhang Zi-Gang, Luo Xiaoyan, Fossey John, Deng Wei-Ping. DDQ-Mediated Oxidative Coupling: An Approach to 2,3-Dicyanofuran (Thiophene). J. Org. Chem., 2014, 79, 1156-1165. (Highlighted by Synfacts 2014, 10(4), 0374.)
28. Wang Zheng-Lin, An Xing-Lan, Ge Li-Shi, Jing-Hai Jin, Luo Xiaoyan, Deng Wei-Ping. DDQ-mediated oxidation of sp3 C-H bond for the direct synthesisof vicinal tricarbonyl compounds. Tetrahedron, 2014, 70, 3788-3792.
27. Li Yi, Cao Li, Luo Xiaoyan, Deng Wei-Ping. The synthesis of 1, 2-diarylindenes via DDQ-mediated dehydrogenative intramolecular cyclization. Tetrahedron, 2014, 70, 5974-5979.
26. Jiang Shanshan, Hu Bin, Yu Xingxin, Deng WeiPing. Fc-PIP Catalyzed Asymmetric Synthesis of cis-2,3-Dihydrobenzofurans. Chin. J. Chem., 2014, 32, 694-698.
25. Ge Li-Shi, Wang Zheng-Lin, An Xing-Lan, Luo Xiaoyan, Deng Wei-Ping. Direct Synthesis of Polysubstituted 2-Aminothiophenes through Cu(II)-Catalyzed Addition/Oxidative Cyclization of Alkynoates with Thioamides. Org. Biomol. Chem., 2014, 12(42), 8473-8479. (Highlighted by Synfacts 2015, 11(1), 0024.)
24. Luo Xiaoyan, Wang Zheng-Lin, Jin Jing-Hai, An Xing-Lan, Shen Zhenlu, Deng Wei-Ping. Copper-catalyzed α-aminoxylation of 1,3-dicarbonyl compounds with 2,2,6,6-tetramethylpiperidine-1-oxyl (TEMPO) via an aerobic oxidative sp3 C-H bond activation. Tetrahedron, 2014, 70, 8226-8230.
2013
23. Wang Wei-Liang, Feng Yu-Lan, Gao Wen-Qiang, Luo Xiaoyan, Deng Wei-Ping. A highly efficient BF3 Et2O-catalysed intramolecular [3+2] cycloaddition for the synthesis of 3,4-dihydrobenzopyrano[3,4-c]pyrazoles. RSC Adv., 2013, 3, 1687-1690.
22. Wang Zheng, Shi Ying, Luo Xiaoyan, Han De-Man, Deng Wei-Ping. Direct synthesis of pyrroles via 1,3-dipolar cycloaddition of azomethine ylides with ynones. New J. Chem., 2013, 37, 1742-1745.
21. Wang Zheng, Luo Shuai, Zhang Shoude, Yang Wu-Lin, Liu Yang-Zi, Li Honglin, Luo Xiaoyan, Deng Wei-Ping. Catalytic Asymmetric Construction of Quaternary a-Amino Acid-Containing Pyrrolidines via 1,3-Dipolar Cycloaddition of Azomethine Ylides to a-Aminoacrylates. Chem. Eur. J., 2013, 19, 6739-6745.
20. An Na, Tian Bo-Xue, Pi Hong-Jun, Eriksson Leif A., Deng Wei-Ping. Mechanistic Insight into Self-propagation of Organo-mediated Beckmann Rearrangement: A Combined Experimental and Computational Study. J. Org. Chem., 2013, 78, 4297-4302.
19. Xu Su-Ying, Hu Bin, Flower Stephen E., Jiang Yun-Bao, Fossey John S., Deng Wei-Ping, James Tony D. Colorimetric enantioselective recognition of chiral secondary alcohols via hydrogen bonding to a chiral metallocene containing chemosensor. Chem. Commun., 2013, 49, 8314-8316.
18. Jin Hui, Liang Lei, Liu Lifeng, Deng Weiping, Liu Jianwen. HDAC Inhibitor DWP0016 Activates p53 Transcription andAcetylation to Inhibit Cell Growth in U251 Glioblastoma Cells. J. Cell. Biochem., 2013, 114, 1498-1509.
2012
17. Liu Hua, Cao Li, Sun Jia, Fossey John S., Deng Wei-Ping. Iron-catalysed Tandem Cross-dehydrogenative Coupling (CDC) of Terminal Allylic C(sp3) to Styrene and Benzoannulation in the Synthesis of Polysubstituted Naphthalenes. Chem. Commun., 2012, 48 (21), 2674-2676.
16. Shi Yu-Hua, Wang Zheng, Shi Ying, Deng Wei-Ping. Facile and Highly Diastereoselective Synthesis of 3-Aminooxindoles via AgOAc-Catalyzed Vinylogous Mannich Reaction. Tetrahedron, 2012, 68, 3649-3653.
15. Li Yi, Du Wenting, Deng Wei-Ping. NHCs-mediated benzoates formation directly from aromatic aldehydes and halides. Tetrahedron, 2012, 68, 3611-3615.
14. Wang Zheng, Han De-Man, Jia Wen-Ping, Zhou Qi-Zhong, Deng Wei-Ping. Reaction-Based Fluorescent Probe for Selective Discrimination of Thiophenols over Aliphaticthiols and Its Application in Water Samples. Anal. Chem., 2012, 84, 4915 -4920.
13. Li Yi, Cao Li, Luo Xiaoyan, Deng Wei-Ping. Highly Substituted Cyclopentenes Formation via a Stereoselective Tandem CDC Reaction and Cyclization. Chin. J. Chem. 2012, 30, 2834-2838.
12. Hu Bin, Meng Meng, Jiang Shanshan, Deng Wei-Ping. Kinetic Resolution of Aryl Alkenylcarbinols Catalyzed by Fc-PIP. Chin. J. Chem., 2012, 30, 1289-1294.
2011
11. Wang Ming, Shi Yu-Hua, Luo Jun-Fei, Du Wenting, Shi Xiao-Xin, Fossey John S., Deng Wei-Ping. Novel N,O-Cu(OAc)2 complex catalysed diastereo- and enantioselective 1,4-addition of glycine derivatives to alkylidene malonates. Catal. Sci. Technol., 2011, 1(1), 100-103.
10. Fan Wen-Yuan, Wang Zheng-Lin, Li Hong-Chang, Fossey John S., Deng Wei-Ping. A straightforward and efficient synthetic access to biologically active marine sesterterpenoids, sesterstatins 4 and 5. Chem. Commun., 2011, 47, 2961-2963.
9. Wang Ming, Wang Zheng, Shi Yu-Hua, Shi Xiao-Xin, Fossey John S., Deng Wei-Ping. A Remarkable N,O-ligand/Cu(OAc)2 Derived Chiral Complex Catalysed exo-Selective and Enantioselective 1,3-Dipolar Cycloaddition of Azomethine Ylides with Alkylidene Malonates. Angew. Chem. Int. Ed., 2011, 50, 4897-4900. (Highlighted by Synfacts 2011, 7(9), 0969.)
8. Liu Li-Feng, An Na, Pi Hong-Jun, Ying Jun, Du Wenting, Deng Wei-Ping. Facile and odorless one-pot process for the synthesis of N-substituted thioamides via TsCl mediated BR of ketoximes. Synlett., 2011, 7, 979-981.
7. Fan Wen-Yuan, Wang Zheng-Lin, Zhang Zi-Gang, Li Hong-Chang, Deng Wei-Ping. Stereoselective synthesis of marine sesterterpenes, 16-deacetoxy-scalarafuran, (+)-scalarolide and their analogs. Tetrahedron, 2011, 67, 5596-5603.
6. Wang Zheng-Lin, Liu Yang, Zhang Zi-Gang, Li Hong-Chang, Deng Wei-Ping. Concise stereoselective synthesis of marine sesterterpene, 16-deacetoxy-12-epi- scalarafuran acetate and its 14-epimer via intramolecular Diels-Alder addition. Tetrahedron, 2011, 67, 6939-6943.
5. Hu Bin, Meng Meng, Fossey John S., Mo Weimin, Hu Xinquan, Deng Wei-Ping. Optically pure bulky (hetero)arylalkyl carbinols via kinetic resolution. Chem. Commun., 2011, 47, 10632-10634. (Highlighted by Synfacts 2011, 7(12), 1341.)
4. Shi Yu-Hua, Wang Zheng, Hu Bin,Wang Ming, Fossey John S., Deng Wei-Ping. A Ferrocenyl-DHIPOH/ Cu(OAc)2 Complex for Diastereo- and Enantioselective Catalysis of The 1,4-Addition of Glycine Derivatives to Alkylidene Malonates. Org. Lett., 2011, 13, 6010-6013.
2010
3. Hu Bin, Meng Meng, Wang Zheng, Du Wenting, Fossey John S., Hu Xinquan, Deng Wei-Ping. A Highly Selective Ferrocene-Based Planar Chiral PIP (Fc-PIP) Acyl Transfer Catalyst for the Kinetic Resolution of Alcohols. J. Am. Chem. Soc., 2010, 132, 17041-17044.
2. Lin Lu, Li Yi, Du Wenting, Deng Wei-Ping. The NHCs-Mediated Cross-Coupling of Aromatic Aldehydes with Benzyl Halides: Synthesis of α-Aryl Ketones. Tetrahedron Lett., 2010, 51, 3571-3574.
1. Pi Hong-Jun, Liu Li-Feng, Jiang Shan-Shan, Du Wenting, Deng Wei-Ping. The facile one-pot synthesis of N-imidoylbenzotriazoles via a Beckmann rearrangement of ketoximes. Tetrahedron, 2010, 66, 6097-6100.
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